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antithrombin III (Neuart)

✓ Approved

Mitsubishi Tanabe Pharma Corporation · SERPINC1 · Cell-based Therapies

What is antithrombin III?

antithrombin III is a cell-based therapies developed by Mitsubishi Tanabe Pharma Corporation. It is approved for therapeutic indications.

Drug Profile

Brand NamesNeuart
CompanyMitsubishi Tanabe Pharma Corporation
Drug ClassCell-based Therapies
Molecular TargetSERPINC1
StatusApproved

Mechanism of Action

Molecular Targets

antithrombin III acts on 1 molecular target:

SERPINC1serpin family C member 1 (ATIII, AT3D)
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Therapeutic Indications

antithrombin III is developed for 1 unique indication across 1 therapeutic area.

Therapeutic AreaConditionPhase
Vascular disordersThrombosis✓ Approved

Related Research Articles

PubMedAnnals of neurology2026-06-09

Monoallelic POLR3A Variants Cause Early-Onset Peripheral Neuropathy.

Ramos Luiza L P LLP, Parmar Jevin M JM, Wijngaard Robin R, Grosz Bianca R BR et al.

Biallelic variants in genes encoding the RNA polymerase III complex (Pol III) cause a spectrum of neurological disorders primarily affecting the central nervous system. Monoallelic variants have been reported in the POLR3B subunit only, associated with neurodevelopmental disorder, epilepsy, and peripheral neuropathy. We describe a novel Pol III-related disorder caused by monoallelic variants in POLR3A and presenting primarily with peripheral neuropathy. We performed clinical and genetic investigation of the affected families. Biophysical characterization of mutant proteins was performed in silico. Immunoblotting, interactomics, and transcriptomics characterization were done in cellular models. We identified 11 patients across 8 unrelated families harboring heterozygous missense variants in POLR3A, occurring de novo or segregating in an autosomal-dominant fashion. The patients presented with an early-onset, progressive sensorimotor peripheral polyneuropathy with intermediate to demyelinating ranges of nerve conduction slowing, occasionally accompanied with neurological or non-neurological features. White matter abnormalities, characteristic for the biallelic Pol III-related disorders, where not observed in the brain magnetic resonance imaging (MRI) evaluations. The neuropathy-associated variants cluster in regions critical for Pol III activity. We observed mis-regulation of individual Pol III targets and global downregulation of tRNA pools in patient-derived cells. This Pol III dysfunction was not due to impaired POLR3A expression, subcellular localization, or subunit interactions. Our findings expand the Pol III-related disease spectrum beyond the known biallelic phenotypes and establish POLR3A as a novel peripheral neuropathy-associated gene. This work highlights a central role of Pol III dysfunction in disease and reinforces the link between tRNA metabolism and peripheral neurodegeneration. ANN NEUROL 2026.

PubMedBMC oral health2026-06-09

Evaluation of PISA, serum IL-12 and IL-18 in stage III periodontitis with and without type 2 diabetes mellitus: a cross-sectional study.

Mangrolia Shefali S, Kolte Rajashri Abhay RA, Kolte Abhay Pandurang AP, Abullais Shahabe Saquib SS et al.

Previous studies have shown a positive association between periodontitis and diabetes mellitus. However, there is a lack of comprehensive data regarding their combined effect on Periodontal inflamed surface area (PISA), serum Interleukin-12 and Interleukin-18. Therefore, the present study aimed to assess PISA, along with serum IL-12 and IL-18 levels, in individuals diagnosed with Stage III Periodontitis, both with and without type 2 diabetes mellitus (T2DM). 79 participants categorized into: Group I comprising 19 periodontally healthy individuals while Groups II and III included 30 patients each with stage III periodontitis without and with T2DM, respectively. Clinical assessments of probing depth (PD), clinical attachment level (CAL), plaque index (PI), gingival index (GI), bleeding on probing (BOP) and periodontal inflamed surface area (PISA) were performed alongside evaluation of serum IL-12 and IL-18 using enzyme linked immunosorbent assay (ELISA). Additionally, blood investigations included fasting blood glucose, 2-hour postprandial glucose, and HbA1c levels were recorded. Patients in Group II and III demonstrated elevated values for all clinical measurements with significant differences between mean PISA values in Group II (254.21 ± 229.21 mm2) and Group III (401.93 ± 517.61 mm2). Additionally, serum IL-12 and IL-18 were found to be comparatively higher in Group III than in Group II. The findings suggest significantly elevated PISA values for Group III patients and greater severity of periodontal disease as compared to the others. Further research is necessary to better understand the interplay between periodontitis and T2DM, particularly focusing on inflammatory biomarkers and PISA. The trial was registered with the Clinical Trials Registry-India (CTRI/2023/06/053653) on 08/06/2023.

PubMedMarine pollution bulletin2026-06-09

Reliability-integrated multi-objective optimization of offshore oil spill mechanical recovery and oily wastewater management.

Deng Wei W, Bakhtavar Ezzeddin E, Mohammadiun Saeed S, Gharahbagh Abdorreza Alavi AA et al.

Efficient offshore oil spill response requires minimizing response time, operational cost, and residual oil while accounting for operational uncertainty caused by equipment aging and failures. In this study, equipment reliability was modeled using Weibull-based failure probabilities linked to service age and integrated into multi-objective optimization. Two reliability-informed frameworks were developed: the three-objective model (R-OPA-III), which implicitly includes failure and maintenance constraints, and the four-objective model (R-OPA-IV), which explicitly optimizes reliability as an additional objective. Both were benchmarked against deterministic models (OPA-II and OPA-III) under a hypothetical large-scale oil spill in western Canada. Compared with OPA-II and OPA-III, R-OPA-III showed superior consistency, with averages of 437 h of total response time, CAD 1.99 M of total operational cost, and 224.4 m3 of total weathered oil volume, the lowest variability (σ = 9.3 h, CAD 0.018 M, and 7.6 m3), and the shortest normalized Euclidean distance to the ideal point (0.786). R-OPA-IV further extended the Pareto front (132 solutions, hypervolume = 0.850), providing broader trade-offs for decision-makers. This flexibility enables timely recovery and reduced environmental risk under uncertainty. Overall, R-OPA-III offers stable performance for general application, while R-OPA-IV supports adaptive planning. These reliability-informed models enhance the practicality and resilience of offshore oil spill response decision-making.

PubMedBMC ophthalmology2026-06-09

Real-world data analysis of cranial nerve III, IV, and VI palsies: demographics, association factors, and comparative all-cause mortality.

Hsu Chia-An CA, Hsu Min-Huei MH, Melisa Septi S, Yen Ju-Chuan JC

Binocular diplopia is a distressing clinical condition that prompts clinicians to investigate underlying etiologies, particularly cranial nerve (CN) III, IV, or VI palsies. These may arise from microvascular ischemia, inflammation, trauma, compression, or neuromuscular junction disorders. This study aims to explore the association factors of these three ocular motor cranial nerve palsies and to compare their respective all-cause mortality rates using the real-world TriNetX Clinical Research Database (TriNetX CRD). TriNetX is a global federated administrative database with real-time updates of electronic medical records (EMRs). We used the US Collaborative Network within the TriNetX platform to establish the patient cohorts. This network contains electronic health record data from more than 100 million patients across 68 US healthcare organizations (HCOs). This study utilized TriNetX platform to analyze the demographics and associated factors of ocular motor cranial nerve palsies, including diabetes, hypertension, acute myocardial infarction (AMI), overweight status, blood glucose and lipid profiles, body mass index (BMI), and history of brain aneurysm surgery, through intergroup comparisons using paired t-tests. All-cause mortality was assessed using Cox proportional hazards modeling and Kaplan-Meier survival analysis. The average age at presentation was 63, 57, and 60 years for CN III, IV, and VI palsies, respectively, with a slight male predominance. CN VI palsy was the most common, followed by CN IV and CN III palsies. CN III and CN VI palsy cohorts were more commonly associated with diabetes, hypertension, AMI, overweight, and brain aneurysm surgery, suggesting a microvascular or compressive etiology. In contrast, the CN IV palsy cohort was younger and more similar to the general population in clinical and laboratory characteristics. Regarding all-cause mortality, the CN III palsy cohort had the poorest survival, followed closely by the CN VI group, while the CN IV group exhibited the most favorable survival outcome. This study confirmed that CN VI palsy is the most frequent cause of ocular motor nerve palsy leading to binocular diplopia. Notably, CN III and VI palsies shared similar vascular and compressive association factors, while CN IV palsy appeared to be more frequently linked to congenital or traumatic origins. These differences were reflected in the mortality analysis, where CN III palsy showed the worst prognosis, CN VI a slightly better but comparable pattern, and CN IV the best survival outcome. Using the TriNetX CRD, this study delineated the demographic profiles, associated clinical factors, and survival outcomes of patients with ocular motor cranial nerve palsies. The typical demographic was males in their late 50s to early 60s, with CN VI being the most frequently affected nerve. CN III and VI palsies were more often associated with microvascular and compressive conditions, which correlated with higher mortality. Conversely, CN IV palsy was associated with a younger population and more benign clinical profiles, reflected in better survival outcomes.

PubMedJournal of children's orthopaedics2026-06-09

Factors associated with open reduction of pediatric type III supracondylar humerus fractures.

Najd Mazhar Farid F, Zareie Bushra B, Shariatzadeh Hooman H, Hasan Ahmad A et al.

Supracondylar fractures of the humerus are the most common elbow fractures in children. Surgical fixation is necessary in cases with complete displacement (Gartland type III), with closed reduction and pin fixation being preferred. It is sometimes impossible. This study examined radiological and clinical factors that influence the selection of open reduction methods for these fractures. A retrospective study was designed to investigate children aged 3-13 years with Gartland type III supracondylar humeral fractures (OTA/AO 13-M/3.1 III) treated with closed and open reduction techniques. We enrolled 140 patients in the closed reduction group (mean age 6.27) and 90 in the open reduction group (mean age 6.86). The main outcomes were achieving adequate closed reduction or switching to open reduction. We used univariate analysis and multivariate logistic regression to find independent risk factors and odds ratios for open reduction and internal fixation. Older children were significantly more likely to have flexion-type fractures (P = 0.001). The final univariate analysis showed that older age (odds ratios (95% confidence interval): 1.1 (1, 1.3)), flexion-type fractures (odds ratios (95% confidence interval): 3.2 (1.4, 7.4)), low-level (below isthmus) fractures (odds ratios (95% confidence interval): 2.2 (1.3, 3.9)), and Pucker sign (odds ratios (95% confidence interval): 2 (1, 4)) were factors that significantly increased the chance of open reduction and internal fixation. The influence of older age and low-level fracture was also strongly demonstrated in multivariate analysis. As age increases, the chance of a flexion-type fracture rises, and thus the chance of needing open reduction. Low-level fractures reduce the possibility of achieving a stable closed reduction by creating a smaller, more cartilaginous distal fragment. Level III.

PubMedOrganic letters2026-06-09

Light-Driven Iron-Mediated Thiotrifluoromethylation of Alkenes Using CF3CO2H.

Zhou Ying-Hui YH, Zhou Ting T, Cheung Chi Wai CW, Ma Jun-An JA

Fluorinated thioethers are important motifs in medicinal and agrochemical chemistry, but modular synthesis of structurally complex derivatives remains challenging. Herein we report a photoinduced iron(III)-mediated thiotrifluoromethylation of alkenes using trifluoroacetic acid as an inexpensive CF3 radical source and S-aryl benzenesulfonothioates as arylthio donors. Under purple-light irradiation, simple iron(III) salts enable a three-component reaction that affords diverse aryl 3,3,3-trifluoropropyl sulfides with broad scope and good functional group tolerance. The products are readily elaborated and applied to late-stage modification of complex molecules, providing a simple and scalable route to fluorinated sulfur-containing scaffolds.

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