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minocycline hydrochloride

✓ Approved

PreCision Dermatology · Small Molecule · Small Molecule

What is minocycline hydrochloride?

minocycline hydrochloride is a small molecule developed by PreCision Dermatology. It is approved for therapeutic indications via oral (po).

Drug Profile

CompanyPreCision Dermatology
Drug ClassSmall Molecule
RouteOral (PO)
StatusApproved

Therapeutic Indications

minocycline hydrochloride is developed for 1 unique indication across 1 therapeutic area.

Therapeutic AreaConditionPhase
Infections and infestationsStreptococcal infection✓ Approved

Related Research Articles

PubMedNeuroprotection (Chichester, England)2026-07-25

Graded traumatic brain injury severity differentially modulates microglial and astrocytic polarization states and response to minocycline.

Yu Yan Y, Wang Chen C, Zhu Jinyu J, Du Jiahui J et al.

Traumatic brain injury (TBI) involves complex secondary injury cascades in which neuroinflammation is a prominent driver. The lack of standardized models capturing a spectrum of injury severities has hindered a systematic understanding of the associated cellular and molecular responses. This study aims to systematically characterize the dynamic responses and phenotypic shifts of neurons, microglia, and astrocytes during the acute and subacute phases following TBI of varying severities. By integrating macroscopic histopathological assessments with microscopic cellular analyses and correlating these with early peripheral biomarker changes, we seek to provide a solid experimental foundation for understanding TBI mechanisms and developing severity-stratified diagnostic and therapeutic strategies. Male mice were randomly assigned using a computer-generated randomization sequence to the following experimental groups: Sham group, mice that underwent only craniotomy (n = 10 per group); Mild group, mice with a 0.5 mm depth impact on the right motor cortex (n = 10 per group); Moderate group, mice with a 1.0 mm depth impact on the right motor cortex (n = 10 per group); Severe group, mice with a 2.0 mm depth impact on the right motor cortex (n = 10 per group). On Days 1, 3, 7, and 14 after injury, tissue damage was assessed using Nissl staining; anxiety-like behavior was evaluated using the elevated plus maze; cognitive function was assessed using the Y-maze test; motor function was evaluated using the open field test, balance beam test, rotarod test, and gait analysis; neuronal apoptosis and glial cell polarization levels were assessed using immunofluorescence staining; and changes in peripheral serum markers were measured using enzyme-linked immunosorbent assay (Elisa). In addition, severely injured mice received minocycline treatment (45 mg/kg, n = 12 per group) from 30 min to Day 3 post-injury, while the control group received the same volume of saline. For comparisons between groups at a single time point, one-way analysis of variance (ANOVA) followed by Tukey's multiple comparisons test was used. For comparisons between groups across multiple time points, two-way ANOVA followed by Tukey's multiple comparisons test was applied. Impact depth was directly correlated with histopathological lesion volume and dictated the trajectory of functional recovery. Motor deficits and neuronal apoptosis scaled with injury severity. The neuroimmune response was severity-dependent: mild TBI triggered a transient, reparative response dominated by M2 microglia and A2 astrocytes. In contrast, severe TBI provoked an early and sustained pro-inflammatory state, characterized by persistent M1 microglial and neurotoxic A1 astrocytic activation (n = 4 per group, p < 0.0001). Furthermore, severe injury led to significant acute elevations in serum interleukin-6 (IL-6) and ubiquitin carboxy-terminal hydrolase L1 (UCHL1) within 6 h post-injury (n = 3 per group, p < 0.0001). Minocycline treatment attenuated neuroinflammation, improved motor function, and promoted a shift in microglial polarization toward the protective M2 phenotype (n > 4 per group, all p < 0.05). Our findings establish that TBI severity is a critical determinant of the post-injury neuroimmune microenvironment, with severe injuries driving a maladaptive, chronic inflammatory response. This graded model provides a robust framework for identifying severity-specific biomarkers and validates the rationale for developing precision immunomodulatory therapies stratified by injury severity.

PubMedInternational journal of pharmaceutics2026-07-25

Development of propranolol hydrochloride extended-release lipid matrix tablets for pediatric use.

Broocks Stefanie S, Gebhardt Melanie M, Klein Sandra S

Although solid oral dosage forms are widely used in adult drug therapy, age-appropriate formulations for pediatric patients remain limited. The development of suitable dosage forms is challenged by specific requirements regarding excipient safety, tablet size, and dose flexibility, as well as the need to improve therapy adherence in the context of frequent dosing. This study aimed to develop a pediatric-appropriate extended-release matrix tablet based on lipid matrix formers, with particular attention to the use of safe excipients and the selection of excipients based on sustainability considerations. Lipid-based excipients, selected due to their natural origin and similarity to dietary fats, were investigated and compared with conventional matrix formers. A formulation screening approach was applied to identify promising candidates based on drug release after one hour, followed by further evaluation of manufacturability, tablet hardness, and extended-release performance. In addition, the influence of a physiological pH-gradient, bile salts, and long-term storage on drug release was assessed. The selected formulations showed good manufacturability, uniformity, and sustained drug release. Overall, several lipid-based matrix formulations suitable for pediatric use were identified, providing a promising basis for the development of solid oral extended-release dosage forms for children.

PubMedFrontiers in immunology2026-07-25

Multifunctional antimicrobial effects of Lactobacillus johnsonii against A/E pathogens Enteropathogenic E. coli and Citrobacter rodentium.

Vasamsetti Sai Madhuri SM, Khaderbad Yasaswi Y, Sarmah Novelina N, Atham Hari Naga Papa Rao HNPR et al.

Enteropathogenic Escherichia coli (EPEC) remains a leading cause of childhood diarrhea in low-resource settings, and escalating antimicrobial resistance necessitates non-antibiotic therapeutic approaches. This study investigates Lactobacillus johnsonii as a probiotic candidate capable of limiting A/E-pathogen colonization and attenuating infection-associated intestinal inflammation. The probiotic properties of L. johnsonii were evaluated through assays of gastrointestinal tolerance, epithelial adhesion, antimicrobial activity, biofilm inhibition, and pathogen exclusion. Secreted antimicrobial activity was investigated by fractionation and untargeted metabolomic profiling. Therapeutic efficacy was further assessed in an antibiotic-perturbed Citrobacter rodentium mouse infection. L. johnsonii exhibited robust gastrointestinal resilience (acid pH 1.5-2.5; 0.3% bile) and strong adhesion to human intestinal epithelial cells. In vitro, live L. johnsonii markedly inhibited EPEC growth, disrupted pre-formed biofilms, and displaced adherent pathogens from epithelial surfaces. In an antibiotic-perturbed Citrobacter rodentium infection model, oral L. johnsonii administration reduced pathogen loads in feces and colonic tissues by 3-4 log units, restored colon length, and alleviated epithelial ulceration and inflammatory infiltration. Mechanistic analyses revealed dual antimicrobial actions: nutrient competition and secretion of low-molecular-weight (<75 kDa) bactericidal factors active at ~30 µg mL-1. Untargeted metabolomic profiling of the active fraction generated putative annotations of chemically diverse small molecules, including fatty-acid and hydroxy-acid class compounds, as well as candidate metabolites such as quinine hydrochloride, aloperine, and γ-glutamylglutamine, thereby providing a foundation for future targeted validation of individual antimicrobial components. Notably, probiotic treatment reduced mucosal neutrophil infiltration and preserved epithelial architecture, suggesting attenuation of infection-associated inflammation. Collectively, these findings support L. johnsonii as a multifunctional probiotic that integrates biofilm disruption, metabolic competition, and immune-protective activity. The study highlights its translational potential as a probiotic-based intervention to manage attaching-and-effacing enteric infections and mitigate antibiotic reliance in vulnerable populations.

PubMedHospital pharmacy2026-07-25

Artificial Intelligence and Large Language Models as Decision-Support Tools in Hospital Compounding Pharmacy: A Proof-of-Concept Study.

Castellana Eleonora E, Chiappetta Maria Rachele MR

To evaluate the efficiency and reliability of a large language model (LLM) as a decision-support tool in hospital compounding pharmacy for pediatric extemporaneous preparations requiring assessment of drug crushability, regulatory compliance, and formulation feasibility. A proof-of-concept study compared a structured LLM-assisted workflow with the traditional manual information retrieval process in a hospital pharmacy setting. The LLM (Claude Sonnet 4.6) was configured with a standardized prompt to extract and consolidate data from multiple authoritative sources: the Friuli Venezia Giulia "Do Not Crush" list, the Italian Medicines Agency (AIFA) database for Summary of Product Characteristics (SmPC), AIFA Law 648/96 off-label use lists, and the Stabilis database for oral liquid formulation stability. Two representative drugs, propranolol hydrochloride and imatinib mesylate, were analyzed. For each drug, the model generated a structured output including crushability, regulatory information, off-label status, and extemporaneous formulation data. The same queries were manually performed by an experienced hospital pharmacist. Primary outcome was information retrieval time; secondary outcomes included completeness and accuracy. The LLM-assisted workflow reduced retrieval time to less than 2 minutes per drug (mean 1 minute 45 seconds), compared with a mean of 20 minutes (range 15-25 minutes) for the manual process, plus an additional 5 to 10 minutes for transcription. Output completeness was 100%, with all predefined fields correctly populated. The model accurately classified drug crushability and correctly identified Law 648/96 regulatory status. For propranolol, the system identified crushability, pediatric off-label authorization, and SyrSpend-based formulations with stability data of up to 146 days at room temperature. For imatinib, the model highlighted cytotoxic handling precautions, identified the absence of SyrSpend formulations, and retrieved alternative formulation stability data (30 days refrigerated). A properly configured LLM can function as an effective decision-support tool in hospital compounding pharmacy, improving efficiency while maintaining high standards of completeness, accuracy, and regulatory compliance. These preliminary results support further investigation into the integration of the LLM system into routine pediatric galenical preparation practice.

PubMedBiomedicine & pharmacotherapy = Biomedecine & pharmacotherapie2026-07-24

Tailoring pH-responsive charge-conversional interfaces in ionizable lipid-based nanoliposomes for synchronized co-delivery and synergistic therapy of triple-negative breast cancer.

Choi Yeji Y, Choung Ki-Hoon KH, Jin Minki M, Yoon Moon Sup MS et al.

Combination chemotherapy is often limited by the distinct physicochemical properties and intracellular behaviors of individual drugs. This limitation leads to poorly coordinated delivery in tumor tissues. In this study, pH-responsive ionizable nanoliposomes were developed using the ionizable lipid DLin-DMA to co-deliver erlotinib and doxorubicin hydrochloride. This approach introduces a novel spatial and temporal synchronization strategy for two mechanistically distinct drugs within a single carrier. The resulting nanoliposomes formed stable nanoscale assemblies with an optimized particle size of 139.8 nm and high encapsulation efficiencies of 84.8% for erlotinib and 80.8% for doxorubicin hydrochloride. The formulation exhibited a pronounced pH-dependent surface charge transition. It remained near neutral under physiological conditions but converted to a cationic state in acidic environments relevant to tumors. This charge conversion triggered a sequential drug release profile, featuring an immediate accelerated release of doxorubicin hydrochloride for rapid cytotoxicity alongside a steady sustained release of erlotinib for prolonged targeted inhibition. In MDA-MB-231 triple-negative breast cancer cells, this coordinated cellular internalization and subcellular distribution resulted in profound synergistic cytotoxicity, which was quantitatively confirmed by a Combination Index of 0.427. In vivo evaluations using an MDA-MB-231 xenograft model further demonstrated that the charge-conversional mechanism significantly enhanced tumor accumulation and deep tissue penetration following systemic administration. This targeted accumulation led to robust tumor growth suppression without pronounced systemic toxicity. Overall, this study demonstrates how ionizable lipid chemistry can orchestrate the intracellular fate of chemically dissimilar small molecule drugs, providing a highly effective materials-based framework for synergistic combination therapy in solid tumors.

PubMedIDCases2026-07-24

Hearing loss as the initial manifestation of Chlamydia psittaci pneumonia in an older adult: A case report and literature review.

Wu Hailing H, Li Mengyuan M, Zhang Yuan Y, Zhang Jinghua J et al.

Chlamydia psittaci (C. psittaci) pneumonia is a zoonotic infection that typically presents with fever, cough, and fatigue. Sudden sensorineural hearing loss is an uncommon manifestation and may lead to early misdiagnosis. We report a 67-year-old woman admitted with fever for 1 week and hearing loss for 3 days. Chest computed tomography revealed extensive consolidation in the right lung, and empirical anti-infective therapy was ineffective. Targeted next-generation sequencing (tNGS) of bronchoalveolar lavage fluid (BALF) detected C. psittaci. Following confirmation of the diagnosis, antimicrobial therapy was switched to minocycline. The patient's temperature normalized, hearing improved significantly, pulmonary lesions regressed, and follow-up chest imaging showed near-complete absorption of infiltrates. This case indicates that C. psittaci pneumonia can initially present with hearing loss. Careful evaluation of avian exposure history, characteristic imaging findings, and early molecular pathogen testing may facilitate timely diagnosis and tetracycline-based targeted treatment.

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