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losartan + HCTZ (Gizaar / Hyzaar / Cozaar plus)

✓ Approved

Merck & Co. · AGTR1 · Small Molecule

What is losartan + HCTZ?

losartan + HCTZ is a small molecule developed by Merck & Co.. It is approved for therapeutic indications via oral (po).

Drug Profile

Brand NamesGizaar, Hyzaar, Cozaar plus
CompanyMerck & Co.
Drug ClassSmall Molecule
Molecular TargetAGTR1, SLC12A3
RouteOral (PO)
StatusApproved

Mechanism of Action

Molecular Targets

losartan + HCTZ acts on 2 molecular targets:

AGTR1angiotensin II receptor type 1 (HAT1R, AT1)
SLC12A3solute carrier family 12 member 3 (NCCT, NCC)
Want deeper analysis?Noah AI can explain complex mechanisms and compare to similar drugs.

Therapeutic Indications

losartan + HCTZ is developed for 1 unique indication across 1 therapeutic area.

Therapeutic AreaConditionPhase
Vascular disordersHypertension✓ Approved

Related Research Articles

PubMedScientific reports2026-05-24

Multi-scale temporal convolution attention network for state-of-charge estimation in Li-ion batteries.

Sulthana S Fouziya SF, Sivaramkrishnan M M, Venkatesan G G, Isaac JoshuaRamesh Lalvani J J

Accurate estimation of the State of Charge (SOC) in lithium-ion batteries is critical for the safety, reliability, and efficiency of energy storage systems and electric vehicles (EVs). The traditional model-based SOC estimation approaches have their limitations when it comes to the issues of battery aging, dynamic load variations, and temperature fluctuations, while the existing deep learning methodologies mostly struggle to capture the short-term transients and long-term SOC evolution at the same time. To address these issues, the present study proposes a Multi-Scale Temporal Convolution Attention Network (MSTCAN), a fusion of multi-scale temporal convolutions for hierarchical feature extraction and an attention-based technique to highlight the most significant signals from voltage, current, and temperature measurements. The data set of Tesla Model-3 2170 Li-ion battery is prepared for processing by the utilization of data cleaning, min-max normalization, and cycle-based segmentation, resulting in enhanced feature quality and temporal representation improvements. An experiment was carried out where the different techniques were compared, and among them, MSTCAN achieving 1.25% Root Mean Square Error (RMSE), 0.97% Mean Absolute Error (MAE), 3.12% max error, and the coefficient of determination (R²) value of 0.998, thus surpassing the traditional and deep learning methods as well. The study's findings affirm both the model's robustness and its reliability, thus providing an attractive solution that could effectively upgrade the performance and even the efficiency of battery management system (BMS) in practical electric vehicle applications.

PubMedCancer treatment reviews2026-05-23

Central nervous system and leptomeningeal metastases in patients with HER2-positive breast cancer: A comprehensive review and therapeutic algorithm proposal.

Caltavituro Aldo A, Buonaiuto Roberto R, Longobardi Alessandra A, Trasacco Paola P et al.

Breast cancer (BC) is the second leading cause of brain metastases (BMs). The incidence of BMs has increased over the last decades as results of both the improvement in imaging detection power and the longer life expectancy of patients with metastatic disease. In human epidermal growth factor receptor 2-positive (HER2 + ) advanced BC, the incidence of BMs is especially high and is associated with poor prognosis. The central nervous system (CNS) has historically been considered a sanctuary site since the blood-brain barrier prevents the penetration of most therapeutic agents. Therefore, loco-regional therapies, such as surgery or radiotherapy, have largely represented the only effective strategies for treating intracranial disease. However, the development of several anti-HER2 agents with proven CNS efficacy has resulted in unprecedented disease control, raising the question of the optimal strategy to adopt in the management of both extracranial and intracranial disease. Here, we provide a comprehensive narrative review of the therapeutic management of HER2 + BMs and leptomeningeal disease, highlighting recent advances in the efficacy of both locoregional and systemic strategies and briefly discuss brain imaging screening and biomarkers for BMs risk stratification. Building on this evidence, we propose an updated, integrated treatment algorithm designed to optimize clinical decision-making.

PubMedMedicine2026-05-23

Post COVID-19 treated with AstraZeneca vaccine exacerbates arthritis with susceptibility to herpes in an older woman: A case report.

Guzman David Calderon DC, Brizuela Norma Osnaya NO, Herrera Maribel Ortiz MO, Peraza Armando Valenzuela AV et al.

Rheumatoid arthritis (RA) is an autoimmune inflammatory disorder that has seriously affected human health worldwide. This report describes a rare case of herpes infection, secondary to RA, that emerged after coronavirus disease 2019 (COVID-19) infection or vaccination. Despite pharmacological intervention for arthritis, herpes, and mental health symptoms, the patient's condition has not improved. A 70-year-old female homemaker, weighing 110 lbs, sought urgent care for persistent dysphoric mood and irritability attributed to a post-COVID infection. The ill-health condition set in with severe pain, followed shortly by the onset of herpetic lesions. She experienced the symptoms while suffering from chronic fatigue syndrome. A diagnosis of arthritis was made at the age of 60, and the patient has since been under treatment with analgesic therapy and prednisone. However, her doctor advised lowering the dose of her RA medications. At the age of 67, she developed herpes. She is currently on acyclovir and remains fully compliant with her medication. A simple skull magnetic resonance study depicted the absence of intracranial abnormality. Electromyography of normal muscles is silent at rest, without neuropathy. Cholesterol, sodium, chlorine, erythrocyte, and eosinophil were at the lower limit of normal, while lipase, phosphatase alkaline, and platelets were at the upper limit. An integrative approach was taken, combining pharmaceutical prescriptions for arthritis, herpes, and mood symptoms with unconventional complementary therapies. Oral food intake was initiated and well-tolerated; however, the patient's clinical condition did not improve with the current treatment. She is currently recovering at home on a regimen of vitamins, acyclovir, and analgesics. While she has shown clinical improvement, some complications have emerged. Diagnostic findings demonstrate that her health is not within normal limits, necessitating a daily regimen of prednisone, analgesic therapy, and hydroxyzine/losartan. This case highlights the importance of studying patients with RA. Risk factors for severe COVID-19 outcomes include older age and comorbidities. This case highlights the potential for COVID-19 infection or immunization to precipitate a flare of preexisting arthritis, causing severe lower limb manifestations and sacroiliitis (low back pain/sciatica) in older individuals receiving management for rheumatic disease. Immune abnormalities in patients treated with prednisone are elements in deciding the prescription and duration of this drug, and a neurological assessment is essential.

PubMedEnvironmental toxicology and pharmacology2026-05-22

Risk of skin cancer from hydrochlorothiazide and other diuretics across races: a global cohort study.

Lee Chaw-Ning CN, Shao Shih-Chieh SC, Yang Chao-Chun CC, Hung Jia-Horung JH et al.

Hydrochlorothiazide (HCTZ) has been linked to increased skin cancer risk. However, comparative evidence across racial groups remains limited. Using TriNetX, a global database, we evaluated the association between thiazide diuretic use and skin cancer risk across whites and other races within a single analytic platform, including both HCTZ and non-HCTZ thiazides. To determine if the skin cancer risk associated with thiazide diuretics varies by racial group. Using the TriNetX platform, we analyzed adults with newly treated hypertension, applying propensity score matching for baseline covariates, and calculated adjusted hazard ratios (aHRs) for skin cancers. Comparing to non-diuretic antihypertensive drug (NDAH) use, HCTZ increased the risk of keratinocyte carcinomas (KC) (aHR 1.40), squamous cell carcinoma (aHR 1.75), basal cell carcinoma (aHR 1.46), and malignant melanoma (aHR 1.37) only in the White population. No increased risk was found in the Asian, Hispanic, or Black populations. Chlorthalidone showed a similar pattern for KC, with increased event rates only in the White population. HCTZ is associated with an increased risk of skin cancers only among whites, while similar associations were not observed in other races. These findings may be considered when prescribing thiazide diuretics in this population.

PubMedThe Journal of chemical physics2026-05-22

Crystallite shape and packing of paramagnetic microcrystalline powders from the measurement and calculation of bulk magnetic susceptibility shifts in solid-state NMR.

Balavoine Gabriel G, Carvalho José P JP, Koppe Jonas J, Pell Andrew J AJ

The size and shape of crystallites strongly influence the properties of functional materials yet remain challenging to access experimentally. In paramagnetic solids, the bulk magnetic susceptibility (BMS) contributes a part to the measured nuclear magnetic resonance (NMR) shift tensor, which depends strongly on particle shape and packing. Here, we use a Fourier-space approach to quantify BMS shifts in LiFePO4 and use the 7Li magic-angle spinning NMR spectra to directly probe the crystallite shape and size. By disentangling internal and external BMS shift contributions from the crystallite of interest and its neighbors, we show that particle shape anisotropy leaves a clear signature in the NMR line shape. Combining BMS modeling with quantum-chemical local shift parameters yields excellent agreement with experimental spectra and enables the extraction of new morphological insights, highlighting solid-state NMR as a quantitative probe of crystallite morphology in paramagnetic materials.

PubMedClinical orthopaedics and related research2026-05-22

Development and Internal Evaluation of EAST-BMS (East Asian Survival Tool for Bone Metastasis Surgery): A Multinational Machine-learning Survival Prediction Model for Patients Undergoing Surgery for Nonspinal Bone Metastasis in East Asia.

Yang Eunkyu E, Lin Hao-Chen HC, Shimomura Seiji S, Lee Jaemin J et al.

Patients undergoing surgery for bone metastases typically have advanced disease, and postoperative survival varies substantially. Accurate survival estimation is important for surgical decision-making and patient counseling. Several prognostic models have been externally validated in East Asian populations, but these tools were originally developed in Western cohorts and do not incorporate region-specific epidemiology or treatment patterns. (1) To develop, internally evaluate, and select a machine learning-based survival prediction model for patients undergoing surgery for nonspinal bone metastases using a multinational East Asian cohort. (2) To compare the performance of the selected model with that of an established Western prognostic tool developed by the Skeletal Oncology Research Group (SORG). (3) To identify which clinical features carried the greatest importance in the new model that we developed. All patients who underwent surgery for nonspinal bone metastases at three tertiary referral centers in the Republic of Korea, Taiwan, and Japan between January 2009 and December 2022 were included. In total, 1045 patients met the inclusion criteria. The median (range) age at surgery was 64 years (19 to 96), 46% (478 of 1045) of patients were female, and the femur was the most common metastatic site (66% [690]). Data for 3-month, 6-month, 1-year, 3-year, and 5-year overall survival were available for 82% (854), 68% (709), 51% (529), 23% (243), and 15% (160) of patients, respectively. The corresponding survival proportions were 84%, 71%, 56%, 36%, and 31%. Data on routinely available clinical, functional, and laboratory variables were collected, and candidate predictors were predefined based on clinical relevance and data availability across institutions. Missing data were < 4% for all variables in each institution and were handled by multivariate imputation by chained equations. We trained four models using different machine-learning algorithms, and the performance of each model was evaluated using leave-one-site-out validation, in which models were trained on data from two institutions and tested on the remaining institution to ensure separation between training and testing data sets. Model performance was assessed using the Concordance Index (C-index; the ability of the model to correctly rank patients according to their expected survival), Brier score (overall prediction error), time-dependent area under the curve (tdAUC; how well the model distinguishes patients with different survival outcomes at specific time points), calibration slope and intercept (agreement between predicted and observed survival), and decision curve analysis (the potential clinical benefit of using the model to guide treatment decisions). The best-performing model was designated as the East Asian Survival Tool for Bone Metastasis Surgery (EAST-BMS) and was compared with the SORG model. To allow a fair comparison, the performance of the SORG model was evaluated on the same held-out test data sets in each iteration of the leave-one-site-out validation, applying the same performance metrics used to select the final model. Gradient boosting survival analysis demonstrated the most favorable overall performance and was selected as the EAST-BMS. The number of outcome events used for model evaluation was 170 at 3 months and 447 at 12 months. The EAST-BMS achieved tdAUC values of 0.81 (95% confidence interval [CI] 0.78 to 0.85) at 3 months and 0.78 (95% CI 0.70 to 0.84) at 12 months, compared with 0.81 (95% CI 0.74 to 0.86) and 0.76 (95% CI 0.67 to 0.83), respectively, for the SORG model, indicating comparable ability to distinguish patients with different survival outcomes. Brier scores were 0.12 (95% CI 0.09 to 0.15) and 0.23 (95% CI 0.17 to 0.28) for EAST-BMS versus 0.14 (95% CI 0.12 to 0.16) and 0.25 (95% CI 0.15 to 0.34) for SORG, indicating lower prediction error in EAST-BMS. Calibration intercepts were -0.08 (95% CI -0.25 to 0.09) versus -1.06 (95% CI -1.26 to -0.86) at 3 months and -0.35 (95% CI -0.49 to -0.22) versus -1.23 (95% CI -1.37 to -1.08) at 12 months, indicating better agreement between predicted and observed survival in EAST-BMS. Decision curve analysis showed wider threshold probability ranges with positive net clinical benefit for EAST-BMS (0.04 to 0.96 versus 0.05 to 0.66 at 3 months; 0.17 to 0.77 versus 0.08 to 0.67 at 12 months), which means that using the EAST-BMS to guide treatment decisions may provide greater clinical benefit than the SORG model. Albumin, Karnofsky performance status, percentage of lymphocytes, and C-reactive protein level were among the most influential predictors. The EAST-BMS, the first multinational machine-learning survival model for patients from East Asia undergoing surgery for nonspinal bone metastases of which we are aware, demonstrated favorable predictive accuracy and clinical utility. This web-based tool may support personalized prognostic assessment and surgical decision-making. It is freely available as a web-based tool at https://bms.east-mskonco.org. Level III, therapeutic study.

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