Drug Database
TE

teriparatide (Xinfutai)

✓ Approved

Shenzhen Salubris Pharmaceuticals Co., Ltd. · PTH1R · Recombinant Proteins

What is teriparatide?

teriparatide is a recombinant proteins developed by Shenzhen Salubris Pharmaceuticals Co., Ltd.. It is approved for therapeutic indications via injectable (others) or subcutaneous injection.

Drug Profile

Brand NamesXinfutai
CompanyShenzhen Salubris Pharmaceuticals Co., Ltd.
Drug ClassRecombinant Proteins
Molecular TargetPTH1R
RouteInjectable (Others), Subcutaneous Injection
StatusApproved

Mechanism of Action

Molecular Targets

teriparatide acts on 1 molecular target:

PTH1Rparathyroid hormone 1 receptor (PTHR, EKNS)
Want deeper analysis?Noah AI can explain complex mechanisms and compare to similar drugs.

Therapeutic Indications

teriparatide is developed for 1 unique indication across 1 therapeutic area.

Therapeutic AreaConditionPhase
Musculoskeletal and connective tissue disordersOsteoporosis✓ Approved

Related Research Articles

PubMedThe AAPS journal2026-09-19

Artificial Intelligence in Pharmaceutical Regulatory Science: Opportunities, Challenges, and Emerging Frameworks.

Lucas Inês I, Sousa João J, Vitorino Carla C

Digital transformation in pharmaceutical regulatory affairs is accelerating as global submissions grow in complexity and traditional document-based workflows reach their limits. Artificial intelligence (AI), particularly natural language processing (NLP), is increasingly being explored to support regulatory data management, document preparation, and decision support activities. This review examines AI adoption across pharmaceutical regulatory science, including initiatives from major regulatory agencies, AI-supported regulatory workflows, and emerging governance and interoperability frameworks. Current applications include document classification, data extraction, Common Technical Document (CTD) support, pharmacovigilance, and predictive analytics. Key implementation challenges, including explainability, traceability, validation, data quality, interoperability, cybersecurity, and Good Practice (GxP) compliance requirements, are critically discussed. The review further examines emerging regulatory data ecosystems and governance frameworks that may support the responsible integration of AI into regulatory processes. Collectively, these developments highlight the potential of AI to support more structured, interoperable, and efficient regulatory systems while maintaining regulatory oversight and accountability. Current evidence suggests that AI implementation has progressed from conceptual research toward early operational deployment. However, robust evidence demonstrating sustained improvements in regulatory performance and long-term operational impact remains limited.

PubMedF1000Research2026-09-19

The Beekeeping Sector of Kazakhstan and Contributions to the Pharmaceutical Industry: Promising Flavonoids with the Pharmacokinetic Properties Via the Computational Evaluations.

Kaya Şeyda Ş, Selamoglu Zeliha Z, Durna Daştan Sevgi S, Gaipov Tulkinzhon T et al.

Bee products are rich sources of bioactive flavonoids with potential applications in nutraceutical and pharmaceutical research. However, differences in the physicochemical and pharmacokinetic properties of individual flavonoids may substantially influence their drug-likeness and bioavailability. This study aimed to characterize the pharmacokinetic, physicochemical, and drug-likeness profiles of four representative flavonoids commonly associated with bee products myricetin, galangin, kaempferol, and quercetin. In silico pharmacokinetic and drug-likeness analyses were performed using the SwissADME web platform. The investigated compounds were evaluated in terms of physicochemical properties, lipophilicity, aqueous solubility, gastrointestinal absorption, blood-brain barrier (BBB) permeability, P-glycoprotein (P-gp) substrate status, and compliance with established drug-likeness rules, including Lipinski, Veber, Egan, and Muegge criteria. All four flavonoids exhibited favorable molecular properties and an identical predicted bioavailability score of 0.55. Galangin, kaempferol, and quercetin showed high predicted gastrointestinal absorption and fully complied with the Lipinski, Veber, Egan, and Muegge drug-likeness criteria. In contrast, myricetin exhibited comparatively lower predicted gastrointestinal absorption, which may be associated with its higher polarity, greater hydrogen-bonding capacity, and elevated topological polar surface area. None of the investigated flavonoids was predicted to penetrate the BBB or to act as a P-gp substrate. Variations in hydroxyl substitution were associated with marked differences in lipophilicity, aqueous solubility, membrane permeability, and overall pharmacokinetic behavior. Among the compounds evaluated, galangin displayed the most balanced physicochemical and medicinal chemistry profile, whereas kaempferol and quercetin also demonstrated favorable characteristics for oral drug development. The findings indicate that flavonoids associated with Kazakhstan bee products possess distinct but generally favorable drug-likeness and predicted pharmacokinetic profiles. In particular, galangin emerged as the most balanced candidate among the compounds examined. Integrating in silico pharmacokinetic assessment with knowledge of bee-product composition may contribute to the scientific evaluation, quality standardization, and value-added utilization of Kazakhstan's apicultural resources, while providing a basis for further experimental investigation of their nutraceutical and pharmaceutical potential.

PubMedFrontiers in microbiology2026-09-19

Mineral-specific effects on humification and bacterial community succession in industrial-scale spent mushroom substrate composting.

Chang Yuan Y, Miao Nannan N, Zhang Yuhan Y, Wei Yuquan Y et al.

Spent mushroom substrate (SMS) is a lignocellulose-rich agricultural by-product whose slow humification can limit the quality and agronomic value of the resulting compost. This study compared four low-cost mineral amendments: shale powder (S), mullite-based soil conditioner (SC), flue-gas desulfurization gypsum (DG), and rare-earth silico-titanate ore powder (TO). Each mineral was added at 10% of SMS dry mass during 40-day industrial-scale composting. Mineral structure, physicochemical properties, humic fractions, dissolved organic matter (DOM) fluorescence components, and bacterial succession were evaluated. Results showed that mineral amendments accelerated pile heating, prolonged the thermophilic phase, and promoted compost humification. Relative to CK, final humic acid (HA) content increased by 20.6, 28.1, 10.7, and 7.9% in S, SC, DG, and TO, respectively, while the humification index (HI) increased by 25.9, 41.5, 14.9, and 16.0%, respectively, highlighting SC as the strongest overall humification response. EEM-PARAFAC analysis revealed mineral-specific DOM transformation patterns: the relative abundance of the highly humified C3 component increased by 9.1 and 17.3% in S and SC, respectively, whereas DG preferentially increased C2 by 18.8%, and TO caused a slight 2.3% decrease in C3 relative to CK. SC increased the relative proportion of the highly humified C3 component by 17.3%, whereas DG increased that of C2 by 18.8% relative to CK. Mineral amendments also reshaped bacterial succession in a stage-dependent manner. SC favored heat-adapted core genera associated with organic matter transformation and humification during the thermophilic and cooling phases, whereas DG and TO exerted stronger selection for maturation-associated Actinomycetota, particularly Nonomuraea. Mantel analysis further revealed significant associations between mineral-induced shifts in the core bacterial community and changes in composting conditions and humification characteristics (Mantel r = 0.323-0.728, FDR-adjusted p < 0.05). These findings demonstrate that mullite-based conditioner provided the most effective enhancement of SMS compost maturity and humification, providing a scientific basis for the targeted selection of low-cost mineral amendments and the valorization of agricultural by-product.

PubMedThe AAPS journal2026-09-19

Investigating the Role of Phenolic Acid Coformers in Enhancing the Physicochemical Properties of Enzalutamide Coamorphous Systems.

Balaga Venkata Krishna Rao VKR, Chatziadi Argyro A, Ridvan Luděk L, Šoóš Miroslav M

Coamorphous systems are gaining interest as an effective formulation strategy to improve the solubility and dissolution of poorly water-soluble drugs. This study investigates the role of phenolic acids as coformers in enhancing the physicochemical properties of enzalutamide (ENZ), a poorly soluble anticancer drug. Five phenolic acids-p-coumaric acid (CMA), ferulic acid (FRA), cinnamic acid (CNA), vanillic acid (VNA), and p-hydroxybenzoic acid (HBA)-were selected based on their glass-forming ability and potential for molecular interactions. Coamorphous systems were prepared and characterized using powder X-ray diffraction (PXRD), modulated differential scanning calorimetry (mDSC), attenuated total reflectance Fourier-transform infrared spectroscopy (ATR-FTIR), and Raman spectroscopy. All coformers successfully induced amorphization, evidenced by halo patterns in PXRD and single glass transition temperatures in mDSC. Spectroscopic analysis confirmed the absence of strong intermolecular bonding, indicating homogeneous mixing. The coamorphous systems exhibited improved solubility across physiological pH conditions and maintained supersaturation for at least four hours under non-sink dissolution testing. These results highlight the potential of phenolic acids as coformers in developing stable, high-performing coamorphous drug systems to enhance the bioavailability of poorly soluble APIs like enzalutamide.

PubMedCureus2026-09-19

An Early Single-Center Case Series Experience With a Recently Introduced Formulation of Inhaled Treprostinil (Yutrepia).

Moore Christopher R CR, Sharma Munish M, Kim Andrew I AI, Ghamande Shekhar S et al.

Treprostinil inhalation powder produced using PRINT technology (LIQ861; delivered via the RS00 Model 8 dry powder inhaler; Yutrepia) is an FDA-approved inhaled treprostinil therapy for pulmonary arterial hypertension (PAH) and pulmonary hypertension associated with interstitial lung disease (PH-ILD). Evidence from the INSPIRE phase 3 open-label study supported long-term safety and tolerability; however, real-world implementation data remain limited. We conducted a retrospective, single-center observational case series of consecutive patients initiated on Yutrepia in routine clinical practice between June and December 2025. Our cohort included group 1, group 3, and mixed group 1 and 3 treated at our Pulmonary Hypertension Center of Excellence. The primary objective of this study was to evaluate the real-world safety and tolerability of Yutrepia, with particular attention to airway-related adverse events (AEs), dose modification, and treatment discontinuation in routine clinical practice. Secondary outcomes included initial and maintenance doses achieved. Additional AEs recorded include dizziness, headache, nausea, hypotension, hypertension, tachycardia, fatigue, and hypoxemia. All data were calculated using a Wilson 95% confidence interval (CI) given the small sample size. Twenty-two patients were included (mean age: 66.4 ± 13.8 years; 16 (72.7%) female patients). PH etiology was group 1 in 13 of 22 patients (59.1%), group 3 in 3 of 22 (13.6%), and mixed group 1 and 3 in 6 of 22 (27.3%). Of the 22 patients, 17 (77.27%) were on background therapy: 11 of 13 patients (84.62%) in group 1, 1 of 3 patients (33.33%) in group 3, and 5 of 6 patients (83.33%) in mixed group 1 and 3. Airway-specific AEs were documented in 8 of 22 patients (36.4%; 95% CI: 19.7%-57.0%). Shortness of breath occurred in 5 of 22 (22.7%; 95% CI: 10.1%-43.4%), cough occurred in 3 of 22 (13.6%; 95% CI: 4.7%-33.3%), and no cases of throat irritation were documented (0.0%; 95% CI: 0.0%-14.9%). Dose modification due to any AE occurred in 9 of 22 patients (40.9%; 95% CI: 23.3%-61.3%), and no patients required dose modification or discontinuation because of airway-related AEs (0.0%; 95% CI: 0.0%-14.9%). Due to the retrospective design, causal attribution of individual events to Yutrepia could not always be established. In this retrospective, single-center case series of Yutrepia, no airway-related dose modifications or discontinuations were documented; however, the 95% confidence interval (0.0%-14.9%) indicates that clinically relevant event rates cannot be excluded given the small sample size. Overall, however, 54.5% of patients experienced an adverse event, 40.9% required dose modification, and 36.4% discontinued treatment because of an adverse event. These findings should not be interpreted as indicating that Yutrepia was broadly well tolerated. The observed frequencies of airway-related adverse events were descriptively lower for some events than those reported in selected previous studies of inhaled treprostinil, but direct comparisons cannot be made because of differences in study populations, designs, follow-up, and adverse event ascertainment. Given the small sample size and retrospective design, these findings are hypothesis-generating, and larger prospective studies are needed to define persistence, tolerability, and longer-term clinical outcomes.

PubMedInfectious diseases of poverty2026-09-19

Territorial inequities in access to essential medicines for neglected tropical diseases in a decentralised European health system: a nationwide assessment in Spain.

Belhassen-García Moncef M, de la Calle-Prieto Fernando F, Del Moral Sánchez José Manuel JM, Alonso-Sardón Montserrat M et al.

Neglected tropical diseases (NTDs) represent an increasing but often overlooked challenge for European health systems owing to international mobility, migration, travel, and climate-related changes in disease ecology. Although effective treatments exist for most NTDs and many are included in the World Health Organization (WHO) Model List of Essential Medicines, their availability in decentralised high-income health systems remains poorly characterised. This study assessed the availability, accessibility, and territorial variability of essential medicines for NTDs across the autonomous communities of Spain and identified the main barriers to equitable access. A nationwide, cross-sectional study was conducted across the 17 autonomous communities of Spain. Data were collected between January and December 2025 through a structured survey of Hospital Pharmacy Services in centres with expertise in tropical medicine and infectious diseases and were complemented by expert clinical validation. Medicines were classified according to commercial status, access pathways, dispensing circuits, and regional availability. Descriptive analyses summarised inter-regional variability from a health systems and policy perspective. Data were obtained for 63 medicines and vaccines, generating 1134 records from all 17 autonomous communities. Twenty-two medicines were commercially available in Spain, whereas 39 required exceptional access mechanisms. Routine stock availability across all centres was reported in only 31.1% of valid records, while 52.8% reported no routine stock and 16.1% restricted availability to reference centres. Joint management by prescribing physicians and hospital pharmacy services was required in 72.1% of access procedures. Marked territorial variability was also observed in dispensing circuits and financing mechanisms, with 47.9% of valid records requiring full out-of-pocket payment and 47.1% involving co-payment. Access to essential medicines for NTDs in Spain remains structurally fragmented and territorially unequal. Strengthening coordinated national pharmaceutical policies is necessary to reduce reliance on exceptional access mechanisms and ensure equitable, timely, and sustainable access to essential medicines in Spain and other decentralised European health systems.

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