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NI

NIK-127

✓ Approved

Kowa · Small Molecule · Small Molecule

What is NIK-127?

NIK-127 is a small molecule developed by Kowa. It is approved for therapeutic indications via unknown.

Drug Profile

CompanyKowa
Drug ClassSmall Molecule
RouteUnknown
StatusApproved

Therapeutic Indications

NIK-127 is developed for 1 unique indication across 1 therapeutic area.

Therapeutic AreaConditionPhase
Gastrointestinal disordersDiarrhoea✓ Approved

Related Research Articles

PubMedComputer methods and programs in biomedicine2026-05-24

CardioRadNet: Cardiac mass diagnosis through integrated segmentation and radiomic analysis.

Ferretti Meri M, Pagliaccia Michele M, Baggiano Andrea A, Lovato Luigi L et al.

Cardiac masses (CMs), though rare, include a wide spectrum of benign and malignant lesions that require distinct therapeutic strategies. Prior studies typically address narrow classification tasks (e.g., thrombus vs tumor) and rely on manually delineated regions. Building on these gaps, we introduce CardioRadNet: the first integrated framework combining deep learning segmentation and radiomics-based classification on contrast-free T1-weighted cardiac MR, designed to differentiate benign from malignant CMs. A total of 127 patients with pathologically confirmed CMs (62 malignant, 65 benign) were included. A segmentation network incorporating point-based guidance was developed for mass delineation. Radiomic features were extracted from both manually and semiautomatically segmented volumes, and two separate radiomics-based classification models were developed accordingly. Feature selection and classifier performance were optimized using a 5-fold cross-validation. The segmentation network achieved a Dice score of 0.78, with 88% of the radiomic features extracted from the semiautomatic ROIs showing good reproducibility (ICC > 0.6) when compared with those derived from manual ROIs. The two models achieved identical balanced accuracy (0.85) and the same number of misclassifications (both used 10 features). Notably, the semiautomated ROI model yielded one fewer false negative, thereby reducing missed malignant cases. CardioRadNet offers a novel, accurate and contrast-free solution for comprehensive CM classification. Unlike prior studies, it includes the full spectrum of CMs and uses semiautomated segmentation for broader clinical applicability. Overall, this approach supports scalable integration into routine CMR workflows as a decision-support tool for early risk stratification and, in turn, improved patient management.

PubMedAnnals of vascular surgery2026-05-24

Tunnel Transposition Versus Lipectomy for Second-Stage Superficialization of Deep Brachiocephalic Arteriovenous Fistulas: A Multicenter Retrospective Study.

Mabrouk Moustafa M, Fouda Ahmed A, Habiba Ahmed A, Elkassaby Mohammed M et al.

Deeply located arteriovenous fistulas (AVFs) pose a major challenge in hemodialysis access, especially in obese patients, where the cephalic vein lies beyond the optimal cannulation depth. Second-stage superficialization techniques such as tunnel transposition and lipectomy are often required, yet comparative data on their effectiveness remain limited.To compare the clinical outcomes of tunnel transposition versus lipectomy for second-stage superficialization of deep brachiocephalic AVFs. This multicenter retrospective study included 127 patients with mature brachiocephalic AVFs and cephalic veins located >6 mm from the skin surface, who underwent superficialization between January 2020 and May 2024. Patients were assigned to tunnel transposition (n = 69) or lipectomy (n = 58) groups. Outcomes included technical success, time to cannulation, complication rates, and long-term patency. Data were analyzed using t-tests, chi-square tests, and Kaplan-Meier survival analysis. Demographics and comorbidities were comparable between groups. The mean post-superficialization vein depth was lower in the tunnel group (2.48 ± 0.34 mm) compared to the lipectomy group (2.71 ± 0.92 mm), though not statistically significant (p = 0.057). Difficult cannulation occurred significantly more often in the lipectomy group (10.34% vs. 1.45%; p = 0.047). Other complications, including hematoma, infection, thrombosis, and postoperative steal syndrome, were similar. Primary and secondary patency rates up to 24 months showed no significant difference between groups. Tunnel transposition and lipectomy are both effective for superficializing deep brachiocephalic AVFs. However, tunnel transposition may reduce the rate of difficult cannulation and may be preferred in patients with severe vein depth or scarring.

PubMedJournal of pediatric psychology2026-05-24

Diabetes-related distress and quality of life in mothers during the adolescent to young adult transition in type 1 diabetes.

Ness Michelle M MM, Saylor Jennifer L JL

The transition to adulthood presents challenges for families managing type 1 diabetes (T1D), yet maternal well-being during this period remains understudied. Guided by family systems theory and the transactional stress and coping model, this study examined relationships among diabetes-related distress, perceived social support, and quality of life (QoL) in mothers of adolescents and young adults (AYAs; ages 15-25) with T1D. Using a cross-sectional, descriptive correlational design, 72 mothers (M age = 48.6 years, 91.7% White, 87.5% married) of AYAs with T1D (M age = 19.4 years) completed validated measures of T1D-specific QoL, diabetes-related distress, and perceived social support. Kendall's tau-b correlations analyzed associations among study variables. Maternal personal distress demonstrated the strongest negative association with T1D-specific QoL (τb = -0.69, p < .001), followed by mother/AYA relationship distress (τb = -0.58, p < .001) and management distress (τb = -0.56, p < .001). All forms of distress showed large negative associations with emotional well-being and moderate to large negative associations with relationship quality. Overall perceived social support was not significantly associated with T1D-related QoL (τb = 0.15, p = .127), though family (τb = 0.18, p = .036) and friend support (τb = 0.21, p = .015) showed small positive associations with emotional well-being and daily activities. Findings demonstrate that maternal diabetes-related distress, particularly personal distress, was significantly negatively associated with QoL during the AYA period. Results highlight the need for routine distress screening, family-based interventions targeting diabetes-specific conflict, and diabetes-specific support resources tailored to this developmental period.

PubMedJournal of microbiology, immunology, and infection = Wei mian yu gan ran za zhi2026-05-24

Performance and reproducibility of Pylori DuoTect® in a high Helicobacter pylori prevalence Latin American population.

Laszkowska Monika M, Warnakulasuriya Kesari K, Trendler Toria T, Corvalan Alejandro H AH et al.

An accurate, rapid, non-invasive test is critically needed for Helicobacter pylori infection, particularly in under-resourced populations at increased risk of gastric cancer. This study compared the performance of Pylori DuoTect® to a spectrum of other tests. Serum samples collected from Chilean adults with gastrointestinal symptoms who had undergone esophagogastroduodenoscopy were tested with the Pylori DuoTect® test for anti-FliD (flagellar hook-associated protein) and anti-CagA (cytotoxin-associated antigen gene A) antibodies, and compared to testing by urease, histology, whole-cell ELISA, CagA ELISA, and H. pylori-NAPPA array. We calculated sensitivity, specificity, and agreement based on Cohen's kappa statistic of the Pylori DuoTect® test to other tests. Based on histology or rapid urease testing, 156 of 300 individuals (52%) were positive for H. pylori. Based on the Pylori DuoTect® test, 70 (45%) were seropositive for FliD, 94 (60%) for CagA, 127 (81%) for either FliD or CagA, and 37 (24%) for both. Sensitivity of either FliD or CagA detection for a positive H. pylori test by histology or urease testing was 81.1% and specificity was 29.2%. The Pylori DuoTect® test had the highest level of agreement with the CagA NAPPA and ELISA tests (81.3-82.0%). The Pylori DuoTect® test showed high sensitivity but low specificity for H. pylori detection compared to histology or urease testing. However, it aligned well with performance of CagA detection. While this assay may hold promise based on ease of use, it requires additional optimization and validation to better define the performance characteristics across diverse, global populations.

PubMedAnnals of hematology2026-05-24

Value of functional iron parameters in diagnostic re-assessment of MPN: refinement of iron-deficiency markers by zinc protoporphyrin (ZPP).

Manz Kirsi K, Kobrosly Myriam M, Crodel Carl C CC, Al-Ali Haifa H et al.

Iron deficiency assessment in myeloproliferative neoplasms is complicated by chronic inflammation, disease-related anemia, and treatment-induced changes in iron handling. We retrospectively analyzed 445 patients with MPN, including 158 with polycythemia vera, 97 with essential thrombocythemia, 44 with prefibrotic primary myelofibrosis, 127 with overt myelofibrosis, and 19 with MPN-unclassifiable, and compared conventional iron parameters with a population-based SHIP cohort of 4420 participants. ZPP was measured in the MPN cohort using quantitative fluorescence spectroscopy. Compared with SHIP, MPN patients had lower hemoglobin and higher ferritin, and the physiological positive correlation between ferritin and hemoglobin observed in SHIP was reversed in MPN patients, with R = 0.27, 95% CI 0.24 to 0.30, p < 0.001 in SHIP versus R = - 0.45, 95% CI - 0.52 to - 0.36, p < 0.001 in MPN. Median ZPP in the MPN cohort was 43.0 µmol/mol heme, with 123 of 445 patients (27.6%) showing ZPP values > 65 µmol/mol heme and 59 of 445 patients (13.3%) showing values > 100 µmol/mol heme. ZPP differed significantly between MPN entities, with median values of 35.0 µmol/mol heme in ET, 49.4 µmol/mol heme in PV, 36.5 µmol/mol heme in pre-PMF, 54.7 µmol/mol heme in overt MF, and 46.0 µmol/mol heme in MPN-U (p < 0.001). ZPP correlated inversely with hemoglobin in MPN patients (R = - 0.26, 95% CI - 0.35 to - 0.16, p < 0.001), whereas its association with ferritin was weak (R = - 0.10, 95% CI - 0.20 to - 0.00, p = 0.045). Among 80 patients with CTCAE grade ≥ 2 anemia, 58 (73%) had ZPP values above the upper limit of normal. In exploratory multivariable analysis, PV, overt MF, and phlebotomy were independently associated with higher ZPP, whereas CRP and time from diagnosis were not. In JAK2-mutated PV versus ET, ZPP was significantly higher in PV (48.5 versus 37.5 µmol/mol heme, p = 0.010), complementing lower transferrin saturation and higher JAK2 variant allele frequency. These data indicate that ZPP provides a functional readout of iron-restricted heme synthesis in MPN, adds information beyond ferritin and transferrin saturation, and may refine diagnostic reassessment and therapeutic monitoring, particularly in PV and overt MF.

PubMedThe FEBS journal2026-05-23

Adipocyte-specific NIK depletion enhances energy metabolism and glucose tolerance in mice.

Ozcan Atakan A, Uslucan Caroline C, Kizilyer Aleyna A, Agca Samet S et al.

Nuclear factor κB (NF-κB)-inducing kinase (NIK) is a critical component of the noncanonical NF-κB pathway and an important regulator of immune response. NIK deficiency causes loss of lymph nodes, disruption of lymphoid organ structure and deficits in B-cell formation and immunoglobulin production. In this study, we generated adipocyte-specific NIK-knockout (Adipo-NIK-KO) mice to study the role of this protein in adipose tissue metabolism. We found that NIK depletion in mouse primary adipocytes potentiates thermogenic capacity without altering the differentiation of these cells. Loss of NIK in adipocytes stimulated Fibroblast growth factor 21 (FGF21)-induced expression of thermogenic genes, including Uncoupling protein 1 (UCP1) and mitochondrial uncoupled respiration. In fact, enhanced browning of subcutaneous fat depots was detected in Adipo-NIK-KO mice, which also had elevated energy expenditure. These mice exhibited improved glucose tolerance and insulin sensitivity and reduced hepatic lipid deposition upon diet-induced obesity. Similarly, inhibition of NIK by a specific small molecule enhanced metabolic rate and glucose homeostasis in obese mice. Therefore, NIK inhibition holds therapeutic potential for reversing glucose intolerance and insulin resistance associated with obesity.

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