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ciprofloxacin (Aceoto / Cetraxal / Cetraxal Otico)

✓ Approved

Laboratorios SALVAT · Small Molecule · Small Molecule

What is ciprofloxacin?

ciprofloxacin is a small molecule developed by Laboratorios SALVAT. It is approved for therapeutic indications via others.

Drug Profile

Brand NamesAceoto, Cetraxal, Cetraxal Otico
CompanyLaboratorios SALVAT
Drug ClassSmall Molecule
RouteOthers
StatusApproved

Therapeutic Indications

ciprofloxacin is developed for 2 unique indications across 2 therapeutic areas.

Therapeutic AreaConditionPhase
Infections and infestationsOtitis externa✓ Approved
Ear and labyrinth disordersExternal ear inflammation✓ Approved

Related Research Articles

PubMedExperimental eye research2026-05-24

A pilot study on the effect of the exoU gene on biofilm formation by a strain of Pseudomonas aeruginosa isolated from microbial keratitis.

Akter Tanzina T, Hoque M Mozammel MM, Urgeya Kuma Diriba KD, Stapleton Fiona F et al.

To investigate the role of the exoU gene in biofilm formation by comparing wild-type and an exoU knockout mutant of Pseudomonas aeruginosa isolated from microbial keratitis (MK). Biofilm formation by nine exoU-positive P. aeruginosa strains from MK was assessed using the crystal violet assay. The strain exhibiting the highest biofilm production was selected for exoU deletion via homologous recombination using the recombineering plasmid pCasPA. Successful deletion was confirmed using exoU-up-F and exoU-down-R primers and exoU gene specific primers. Cytotoxicity of the wild-type and mutant strains was compared in human corneal epithelial cells using MTT assay. Changes in biofilm between wild-type and mutant strains were assessed using crystal violet assays and confocal laser scanning microscopy. Biofilm-associated antibiotic tolerance was assessed by treating pre-formed biofilms of the wild-type and exoU mutant strains with ciprofloxacin and levofloxacin, followed by quantification of surviving bacteria. PA169 P. aeruginosa produced the highest biofilm amount (OD570/OD660 nm = 2.2 ± 0.15) among the tested strains, and the exoU gene was subsequently deleted from this strain. Biofilm formation was significantly reduced in the mutant (OD570/OD660 nm = 1.4±0.08) compared to its wild-type counterpart (OD570/OD660 nm = 2.2 ± 0.15, p<0.01). Confocal laser scanning microscopy confirmed a decrease in biofilm thickness in the mutant strain relative to the parent strain (8.33 ± 0.58 μm vs 11.67 ± 0.58 μm, respectively, p<0.01). Biofilm-associated antibiotic tolerance was also reduced in the exoU mutant, which showed significantly lower survival than the wild-type strain after exposure to ciprofloxacin at 1× MIC (66.87 ± 4.46% vs 88.38 ± 10.09%) and 10× MIC (49.47 ± 6.36% vs 73.74 ± 7.63%), and levofloxacin at 4× MIC (55.29 ± 14.14% vs 79.80 ± 12.25%) and 20× MIC (12.63 ± 1.59% vs 38.13 ± 3.06%) (all p ≤ 0.03). Additionally, the mutant produced lower cytotoxicity than the wild-type (OD570 8.2±0.23 vs 2.1±0.25, p <0.01). This pilot study suggests that the exoU gene may be associated with biofilm formation and biofilm-associated antibiotic tolerance in the PA169 strain. However, these findings are based on a single clinical strain, and no complementation assay was performed to rule out polar effects of the gene knockout. Further experimental work, including knockout of additional strains, complementation, and strand-specific transcriptomic analysis, is needed to determine whether the observed phenotypic changes are directly caused by deletion of the exoU gene.

PubMedChemistry, an Asian journal2026-05-24

Nature-Inspired Hybrid Photocatalytic System for Degradation of Persistent Organic Pollutants, Including Pharmaceutical Remains Using Solar-Driven Continuous Flow Reactor.

Jaswal Shubham S, Devi Renu R, Singh Anoop A, Kaur Navneet N et al.

Sunlight-driven photocatalytic reactors for wastewater treatment have become a growing hot topic among researchers owing to their inexpensiveness, scalable potential, and minimal ecological impact. Herein, we have utilized 3D printing to fabricate a packed bed reactor (PBR) consisting of an open serpentine channel packed with zinc oxide nanoparticles (ZnO) coated onto silica nanoparticles (SiO2) incorporated on cellulose nanocrystals (CNC) that is ZnO@SiO2@CNC. This developed PBR overcomes the expensive and time-consuming limitations of batch reactors with continuous flow mass treatment of persistent organic pollutants, including methylene blue (MB), Congo red (CR), and ciprofloxacin (CIP). The PBR exhibits remarkable removal efficiency that is further enhanced with increasing turbulence, reaching 99% and 98% for MB and CR, respectively, in just 20 min. Moreover, its potential for the photocatalytic degradation of the CIP antibiotic drug was confirmed with a removal efficiency of 81% in 110 min. The hybrid system was further explored for single-run operation and showed a degradation capacity of 99% for both MB and CR. The nanocomposite applicability to degrade these dyes at different pH levels and degradation pathways was also analyzed. Additionally, similar performance in degrading these persistent pollutants spiked in tap and river water confirmed its environmental applications for real samples.

PubMedJournal of ophthalmic inflammation and infection2026-05-24

Endophthalmitis caused by gram-negative bacteria: etiologies, antibiotic susceptibilities, and treatment outcomes.

Pham Brandon B, Zhang Charles C, Sanchez Victor V, Flynn Harry W HW et al.

To report the etiologies, antibiotic susceptibilities, and treatment outcomes of patients with culture-proven endophthalmitis associated with gram-negative organisms. A single-center retrospective chart review of patients with positive vitreous cultures for gram-negative organisms who presented to a referral center from January 2014 to May 2025. The study included 46 patients (mean age 69.5 years; 58.7% male). The most common isolates were Pseudomonas aeruginosa (19/46, 41.3%), Haemophilus influenzae (8/46, 17.4%), Klebsiella pneumoniae (3/46, 6.5%), Morganella morganii (3/46, 6.5% and Serratia marcescens (3/46, 6.5%). The most common etiologies were post-operative (20/46, 43.5%), followed by bleb-associated (9/46, 19.6%), corneal ulcer (6/46, 13.0%), trauma (5/46, 10.9%), endogenous (4/46, 8.7%), and suture-related (2/46, 4.3%). Most tested organisms were susceptible to amikacin (32/34, 94.1%), gentamicin (33/36, 91.7%), ceftazidime (36/37, 97.3%), tobramycin (33/35, 94.3%), and ciprofloxacin (34/37, 91.9%). Lower susceptibility rates were observed for trimethoprim-sulfamethoxazole (12/18, 66.7%) and ceftriaxone (13/15, 86.7%). All tested organisms were susceptible to meropenem (30/30, 100%). At the last follow-up, only 13.0% (6/46) of patients had a visual acuity of 20/800 or better, and 30.4% (14/46) of patients had no light perception. Enucleation or evisceration was performed in 28.3% of patients (13/46). In the current study, there were generally favorable susceptibilities to commonly used intravitreal antibiotics, but overall patients had poor visual outcomes regardless of specific causative organisms and etiologies. Despite appropriate treatment with intravitreal antibiotics and/or pars plana vitrectomy, enucleation and evisceration were common.

PubMedThe Journal of infection2026-05-24

Health inequalities in Escherichia coli bacteraemia and associated antibiotic resistance: a national surveillance study, England, 2018/19 to 2023/24.

Chudasama Dimple Y DY, Nsonwu Olisaeloka O, Pollington Timothy M TM, Amin-Chowdhury Zahin Z et al.

Health inequalities in Escherichia coli bacteraemia are increasingly recognised, with disadvantaged and minority groups disproportionately affected. Understanding intersecting inequality factors will clarify the poorly understood drivers of overall and resistant E. coli infections. We retrospectively analysed English surveillance data (2018/19-2023/24) of E. coli bacteraemia and resistance. Multivariable logistic regression assessed healthcare- vs community-associated (HA vs CA) and resistant vs susceptible cases. Between April 2018 and March 2024, 242,604 cases of E. coli bacteraemia were reported. Minority ethnic groups were disproportionately represented among patients aged <75 years, in both HA and CA categories. CA cases in females aged 30-44 were 2.7, 4.2, 4.4 and 4.0 times greater in Asian, Black, Mixed and Other ethnicities vs their White counterparts. Multivariable analysis showed odds of antibiotic resistant E. coli bacteraemia were more than twice that in the Asian (OR 2.45, p<0.0001), and 51.0% greater in the Black (p<0.0001) ethnicities, respectively, compared to their White counterparts. Odds of resistance amongst the Asian ethnic group was twice the national average for 2nd (37.2 vs 18.3%) and 3rd generation cephalosporins (35.2 vs 16.1%) and ciprofloxacin (37.1 vs 17.9%). Residing within a care home more than doubled the odds of resistant infection (OR 2.28, p<0.0001). Younger individuals of ethnic minorities particularly females experienced a disproportionate burden of infection, with resistance to key antibiotics particularly elevated in the Asian population. Care home residents had significantly higher rates of CA and resistant E. coli bacteraemia. Greater understanding of the source of infection in these groups is essential to inform targeted interventions.

PubMedChemphyschem : a European journal of chemical physics and physical chemistry2026-05-22

Enhanced Solvation of Hydrophobic Molecules in Aqueous Cygnet Mixtures Explored Through Their Solubility Isotherms.

Lynch Julie J, Sherwood James J, De Bruyn Mario M, Shimizu Seishi S

Herein, we report the apparent aqueous solubilization of acetylsalicylic acid, ciprofloxacin, quercetin, thiabendazole, and vanillin in the presence of a solubilizer, the dioxolane Cyrene derivative, Cygnet. To understand its driving force (i.e., the competitive interactions) within the ternary analyte-Cygnet-water mixtures, experimental data is fit to quadratic solubility isotherms derived recently from statistical thermodynamic fluctuation theory. The insights from the solubility isotherm parameters are (i) attractive Cygnet-analyte preferential interaction for solubilization and (ii) Cygnet-Cygnet self-interaction around the analyte that distinguishes weak synergistic or cooperative solubilization mechanisms. A preferential interaction exists between Cygnet-analyte for all analytes, with synergistic solvation observed for acetylsalicylic acid, ciprofloxacin, thiabendazole, and vanillin; here, maximum, normalized, enhanced solubility increases with analyte hydrophobicity, with thiabendazole experiencing the largest enhancement (17×) and ciprofloxacin the lowest (2.3×). Quercetin undergoes apparent cooperative hydrotropy and displays the largest solubility enhancement overall (41×). Despite these mechanistic differences, analyte-dependent solvation behavior for all analytes can be understood through the same theoretical principle.

PubMedCell chemical biology2026-05-22

SpsB is a target of SOS-response inhibitor OXF-077 and regulates quinolone resistance emergence.

Bradbury Jacob D JD, Walsh Timothy R TR, Lanyon-Hogg Thomas T

Antimicrobial resistance (AMR) is a global health threat, urgently requiring novel compounds with new targets. One emerging strategy is the development of antibiotic adjuvants that inhibit the mutagenic SOS response in bacteria, thus prolonging antibiotic efficacy. OXF-077 is a potent SOS-response inhibitor that suppresses the emergence of ciprofloxacin resistance in Staphylococcus aureus; however, the cellular target of OXF-077 is unknown. We report here the use of affinity-based protein profiling to identify signal peptidase IB (SpsB) as a target of OXF-077. Genetic and chemical studies demonstrated that SpsB is required for the upregulation of the SOS response gene recA and increased frequency of resistance to ciprofloxacin. SpsB is therefore postulated to regulate the SOS response in S. aureus, representing a cell surface peptidase that can be targeted by small molecules to slow the evolution of resistance. Collectively, this work delivers SpsB as an attractive target to combat the urgent threat of AMR.

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