Drug Database
AS

AS0-3B (AS03B1 / AS03B)

✓ Approved

GSK · therapeutic agent

What is AS0-3B?

AS0-3B is a therapeutic agent developed by GSK. It is approved for therapeutic indications via injectable (others) or intramuscular (im) injection.

Drug Profile

Brand NamesAS03B1, AS03B
CompanyGSK
RouteInjectable (Others), Intramuscular (IM) Injection
StatusApproved

Therapeutic Indications

AS0-3B is developed for 1 unique indication across 1 therapeutic area.

Therapeutic AreaConditionPhase
Surgical and medical proceduresOral appliance application✓ Approved

Related Research Articles

PubMedRSC advances2026-07-25

Synthesis and in vitro antiproliferative activity of dolutegravir derivatives against hepatocellular carcinoma via apoptosis-related mechanisms.

Hou Xixi X, Huang Mengmeng M, Zhang Qingqing Q, Yao Qiyan Q et al.

Drug repurposing through structural modification of marketed drugs is a well-established strategy for the discovery of novel therapeutic agents, benefiting from known safety profiles and clinical relevance. Dolutegravir, a widely used HIV integrase inhibitor featuring a nitrogen-oxygen heterocycle, provides an attractive scaffold for exploring new pharmacological activities. In this study, a series of novel dolutegravir derivatives bearing 1,2,3-triazole moieties were synthesized via click chemistry and evaluated for their antitumor activity against hepatocellular carcinoma (HCC). Among them, compounds 3b and 3i exhibited potent antiproliferative activity against HepG2 cells, with IC50 values of 7.89 µM and 15.07 µM, respectively. Both compounds also showed significant inhibitory activity against Huh7 cells, with IC50 values of 2.94 µM for 3b and 4.69 µM for 3i. Further biological studies demonstrated that compounds 3b and 3i significantly induced apoptosis in HepG2 cells, inhibited cell migration in wound-healing assays, and suppressed colony formation. Mechanistic investigations in Huh7 cells further revealed that compound 3b induced concentration-dependent cell death and apoptosis, accompanied by enhanced autophagy and DNA damage. These antitumor effects were associated with significant alterations in apoptosis- and migration-related protein expression. Collectively, these findings demonstrate that dolutegravir-based 1,2,3-triazole derivatives possess promising anti-hepatocellular carcinoma activity and identify compound 3b as a potential lead candidate for further anticancer drug development.

PubMedWorld journal of surgery2026-07-25

Predicting Postoperative Complications in Patients Undergoing Surgery for Inflammatory Bowel Disease.

Lin Viviane V, Pachler Frederik Rønne FR, Pedersen Torben T, Poulsen Jacob Kvist JK et al.

Complications after surgery for inflammatory bowel disease (IBD) have serious short- and long-term consequences. Identifying patients at increased risk may improve outcomes. We utilized a database for patients undergoing surgery for IBD at three Danish hospitals (2017-2022). Stepwise elimination was used to fit a multivariable logistic regression model to predict the occurrence of a Clavien-Dindo postoperative complication ≥ 3B. Patients undergoing resections for Crohn's disease at another Danish hospital (2010-2020) were used for external validation. Additionally, disease-specific models were created. Predictive performance was assessed using measures of discrimination and calibration and clinical utility was assessed using decision curve analysis. A total of 788 patients underwent bowel resection, stoma takedown or restorative proctocolectomy with ileal-pouch-anal anastomosis, with 140 (17.8%) developing a complication. Sex, ASA score, performance status, alcohol intake, diabetes, psychiatric comorbidity, preoperative systemic steroid use, and prior surgery for IBD were identified as predictors in the final model. Discrimination was modest (c-statistic 0.66, Brier score 0.13, AUPRC 0.38). In external validation of 82 Crohn's disease resections, discriminatory performance was comparable (c-statistic 0.66, Brier score 0.14, AUPRC 0.24). Disease-specific models demonstrated improved performance (Crohn's disease: c-statistic 0.74, Brier score 0.11, AUPRC 0.39; ulcerative colitis: c-statistic 0.73, Brier score 0.14, AUPRC 0.49). Predictive performance of a general model was inferior to disease-specific models and insufficient for clinical use, and validation across the full spectrum of IBD resections, is needed to ensure generalizability. However, the model identified factors associated with postoperative morbidity, which may represent targets for prospective studies.

PubMedMolecular neurobiology2026-07-24

Functional and Transcriptional Downregulation of Glutamate Transporters (EAAT1 and EAAT2) via DNMT3B Overexpression in Glial Cells.

Loaeza-Loaeza Jaqueline J, Rodríguez-Campuzano Ada G AG, Hernández-Kelly Luisa C LC, Hernández-Sotelo Daniel D et al.

Glutamate (Glu) is the major excitatory neurotransmitter amino acid in the vertebrate brain. It elicits its actions through the activation of specific receptors in neurons and glial cells. Excitatory amino acid transporters 1 and 2 are the Glu transporters expressed in glial cells, responsible for recycling Glu and executing a protective role against excitotoxicity and neurodegeneration. In neurogenerative diseases and gliomas, glial cells fail to maintain Glu-glutamine homeostasis, triggering excitotoxicity and DNA methylation profile disruption. The aim of this contribution was to investigate the relationship between the methylation gained by DNA methylase 3B overexpression and the functional effect and the expression levels of Glu transporters in glial cell models. First, we confirmed the differential expression and deregulation of excitatory amino acid transporters 1 and 2 in cancer and neurodegenerative diseases. Next, Müller retinal cells were transfected with a DNA methylase 3B vector, and global 5-methylcytosine increased was detected after 48 h. Using a [3H]-D-Aspartate uptake assay in Müller glia cells and the tumoral U87 cells, we determined that de novo methylation affects the functional activity of the Glu transporters. The overexpression of DNMT3B also decreases the expression of Glu transporters in both cell models. Finally, due to the structural characteristics related to methylation deposition in DNA, we analyzed the methylation status of the excitatory amino acid 2 promoter, and we confirmed that DNA methylation increased in U87 cells by the DNMT3B overexpression. These findings suggest that de novo DNA methylation regulates the expression of glial Glu transporters and affects their functional role under excitotoxic environments. This work highlights the DNA methylation mechanism as a promising approach to understand the physiopathology landscape related to excitotoxic processes involved in brain diseases.

PubMedThe Lancet. Neurology2026-07-24

Tolerability, safety, and efficacy of atogepant versus topiramate in adults with migraine (TEMPLE): a randomised, head-to-head, phase 3b trial.

Reuter Uwe U, Dycke Annelies Van AV, Versijpt Jan J, Holle-Lee Dagny D et al.

Oral calcitonin gene-related peptide (CGRP) receptor antagonists such as atogepant have been approved for preventive treatment of migraine but have not been compared directly with conventional oral non-specific preventive treatments. Topiramate is a widely used conventional oral non-migraine-specific preventive treatment for migraine but its use is often limited by poor tolerability. We aimed to evaluate the tolerability, safety, and efficacy of atogepant versus topiramate in adults with migraine, to provide direct comparative evidence to help inform treatment selection. TEMPLE was a phase 3b, randomised, double-dummy, active-controlled trial with a 24-week double-blind treatment period and a 52-week open-label treatment period, done in sites with experience in diagnosing and treating migraine across 12 countries (Austria, Belgium, Canada, Czechia, France, Germany, Hungary, Israel, Italy, Poland, Portugal, and the UK). Participants had a history of migraine and at least 4 migraine days per month on average across the 3 months before screening and during the combined screening and baseline period. Participants were randomly assigned 1:1 to atogepant (60 mg once daily) or topiramate (highest tolerated dose of 50 mg/day, 75 mg/day, or 100 mg/day) using interactive response technology. The primary endpoint assessed tolerability by measuring treatment discontinuation owing to treatment-emergent adverse events during the double-blind period in the safety population (all participants who received ≥1 dose of the study treatment during the double-blind period). Secondary efficacy endpoints related to clinical efficacy were at least 50% reduction from baseline in mean monthly migraine days and change from baseline in mean monthly migraine days during months 4-6 in the modified intention-to-treat population (all randomised participants who received ≥1 dose of study treatment, had an evaluable baseline period of eDiary data, and had ≥1 evaluable postbaseline 4-week [1 month] period of eDiary data within 24 weeks after first dose of study medication [month 1 to month 6], regardless of whether on study treatment or off study treatment). TEMPLE is registered with ClinicalTrials.gov (NCT05748483) and EU Clinical Trials Register (2022-501172-25-00); the double-blind period is completed and the open-label period is ongoing. Between Oct 7, 2023, and April 28, 2025, 730 participants were screened, 545 were randomly assigned, and 540 (479 [89%] female and 61 [11%] male, 517 [96%] White) were included in the safety population (atogepant n=273; topiramate n=267). Discontinuation due to treatment-emergent adverse events across the 24-week double-blind period was lower in the atogepant group (33 [12%] of 273) compared with the topiramate group (79 [30%] of 267; relative risk [RR] 0·4, 95% CI 0·3 to 0·6; p<0·0001). Treatment-related adverse events were reported by 153 (56%) of 273 participants in the atogepant group and 208 (78%) of 267 in the topiramate group. Serious treatment-emergent adverse events occurred in six participants on atogepant and in three participants on topiramate. One serious treatment-emergent adverse event (anaphylactic reaction in the atogepant group) was considered related to study drug. No deaths occurred. More participants experienced at least 50% reduction in mean monthly migraine days in the atogepant group (64% [173 of 270]) compared with the topiramate group (39% [101 of 257], RR 1·6, 95% CI 1·4 to 2·0, p<0·0001) and reduction from baseline in mean monthly migraine days was greater in the atogepant group (least squares mean -6·3 [SE 0·3]) than the topiramate group (-4·5 [0·3]; treatment difference -1·8 [-2·5 to -1·0]; p<0·0001). Atogepant 60 mg once daily showed better tolerability and efficacy across 24 weeks compared with topiramate. Although both topiramate and atogepant are established as effective oral migraine preventive treatments, their usefulness in clinical practice hinges on patients' ability to tolerate treatment. Our findings provide direct comparative evidence that might guide clinicians in selecting the most appropriate preventive therapy for their patients. AbbVie.

PubMedFrontiers in cellular and infection microbiology2026-07-23

Foot-and-mouth disease virus non-structural protein antibody detection: from DIVA serology to repeated-epitope design and multi-species field surveillance.

Bai Yang Y, Gao Kaili K, Wang Siqi S, Cheng Shuchang S et al.

Surveillance for foot-and-mouth disease (FMD) in vaccinated populations requires tests that distinguish vaccine-induced immunity from infection-associated exposure. Structural protein antibodies help assess vaccine response and serotype-specific protection, whereas antibodies to foot-and-mouth disease virus (FMDV) non-structural proteins (NSPs) support DIVA (differentiating infected from vaccinated animals) interpretation only when vaccine purity and vaccination history are considered. Residual NSPs in incompletely purified vaccines, repeated vaccination, antibody kinetics, host species and assay cut-offs all influence interpretation. This Mini Review examines NSP antibody detection based on 3ABC, 3B/VPg repeated-epitope design, complementary NSP targets, competitive or blocking ELISA, multi-species-compatible assays and emerging field-deployable formats. It does not rank platforms as universally superior; instead, it considers reported performance, validation context and field setting. NSP serology is most useful when combined with vaccination records, structural protein serology, RT-qPCR and epidemiological investigation. It can flag possible subclinical exposure or post-outbreak risk, but it is not a standalone test for current shedding, persistent infection or carrier status.

PubMedFrontiers in psychology2026-07-23

When leadership turns covert: conceptualizing and developing a scale for Leader's Manipulative Workplace Behavior.

Luo Dongying D, Wang Zheyuan Z

This research conceptualizes and operationalizes Leader's Manipulative Workplace Behavior (LMWB)-defined as a leader's conscious attempt to alter a subordinate's perception of reality and self-concept to achieve mental control and fulfill selfish goals. A scale measuring the LMWB was developed and validated through multiple empirical samples. In Study 1, items were developed, and their content validity was assessed through two samples of subject matter experts. In Study 2, following item analysis and an initial exploratory factor analysis (EFA) on Sample 2a (N = 249), a 10-item scale was developed. Subsequently, Sample 2b (N = 695) was used in the second EFA to verify the validity of the retained items. In Study 3, Sample 3a (N = 200) was used for confirmatory factor analysis (CFA) and reliability testing, and Sample 3b (N = 256) was used to assess convergent validity, discriminant validity, nomological network, predictive validity, and incremental validity. The results confirmed the scale's reliability and validity and demonstrated that LMWB uniquely predicts employee outcomes beyond the effects of abusive supervision and exploitative leadership. This study provides the first measurement tool for this covert form of psychological manipulation and discusses its significant theoretical and practical implications.

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